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Issue Date
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2020-04-05
Mo(VI) complex catalysed synthesis of sulfones and their modification for anti-HIV activitie
Sah, Ajay Kumar
;
Murugesan, Sankaranarayanan
2020
Glycogen Synthase Kinase 3 (GSK3): Its Role and Inhibitors
Jadhav, Hemant R.
2020
Design, Synthesis and In Vitro Evaluation of 2-Oxo-N-substituted Phenyl-2H-chromene-3-carboxamide Derivatives as HIV Integrase Strand Transfer Inhibitors
Jadhav, Hemant R.
2020
Synthesis and anti-HIV Evaluation of substituted Indole-3-carbaldehyde derivatives
Jadhav, Hemant R.
2020
Study of arginine mimetic benzamidine urea derivatives as PAD4 inhibitors
Jadhav, Hemant R.
2020-09
Pharmacophore based virtual screening, molecular docking, molecular dynamics and MM-GBSA approach for identification of prospective SARS-CoV-2 inhibitor from natural product databases
Murugesan, Sankaranarayanan
2020-12
Targeting a conserved pocket (n-octyl-β-D–glucoside) on the dengue virus envelope protein by small bioactive molecule inhibitors
Murugesan, Sankaranarayanan
2020-10
In-vivo and in-silico toxicity studies of daidzein: an isoflavone from soy
Murugesan, Sankaranarayanan
2020
Leishmaniasis is the most widespread pathogenic disease in several countries. Currently, no effective vaccines are available, and the control of Leishmaniasis primarily relies on decade-old chemotherapy. The treatment for the Leishmaniasis is not up to the mark. Current therapy for Leishmaniasis is ancient and requires hospitalization for the administration. These medications are also highly toxic and resistant. β-carboline, a natural indole containing alkaloid, holds a vital position in the field of medicinal chemistry with a diversified pharmacological action. The current review focuses mainly on the anti-leishmanial effects of β-carboline analogs and their synthetic strategies, structural activity relationship studies (SAR). The past ten years alterations unveiled by β-carboline analogs present in phytoconstituents and various derivatives of synthesized analogs with the mechanism of action were briefly shortlisted and illustrated
Murugesan, Sankaranarayanan
2020-09
Review article| Volume 6, ISSUE 9, e04916, September 2020 PDF [2 MB] Figures Save Share Reprints Request Recent evolution on synthesis strategies and anti-leishmanial activity of β-carboline derivatives – An update
Murugesan, Sankaranarayanan
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Jha, Prabhat Nath
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